Consorzio Interuniversitario per lo sviluppo dei Sistemi a Grande Interfase
Center for Colloid and Surface Science

PUBLICATIONS

Here you can find the updated list of all the publications of CSGI members and affilated staff. Please note that the only publications listed here are those published after the affilation of each member. If you are interested in the whole bibliography of CSGI members, including articles and books published before affilation to CSGI, please refer to academic research databases, such as Scopus, Web Of Science, Google Scholar, ect.

You can use the search bar below to filter the publication list.

2023

1,2,3-Benzoxathiazine-2,2-dioxides - effective inhibitors of human carbonic anhydrases

- Ivanova J. - Abdoli M. - Alessio Nocentini - Žalubovskis R. - Claudiu Supuran
Journal of enzyme inhibition and medicinal chemistry

3H-1,2-Benzoxaphosphepine 2-oxides as selective inhibitors of carbonic anhydrase IX and XII

- Pustenko A. - Balašova A. - Alessio Nocentini - Claudiu Supuran - Žalubovskis R.
Journal of enzyme inhibition and medicinal chemistry

The International Natural Product Sciences Taskforce (INPST) and the power of Twitter networking exemplified through #INPST hashtag analysis

- Singla R.K. - De R. - Efferth T. - Mezzetti B. - Sahab Uddin M. - Sanusi - Ntie-Kang F. - Wang D. - Schultz F. - Kharat K.R. - Devkota H.P. - Battino M. - Sur D. - Lordan R. - Patnaik S.S. - Tsagkaris C. - Sai C.S. - Tripathi S.K. - Găman M.A. - Ahmed M.E.O. - González-Burgos E. - Babiaka S.B. - Paswan S.K. - Odimegwu J.I. - Akram F. - Simal-Gandara J. - Urquiza M.S. - Tikhonov A. - Mondal H. - Singla S. - Lonardo S.D. - Mulholland E.J. - Cenanovic M. - Maigoro A.Y. - Giampieri F. - Lee S. - Tzvetkov N.T. - Louka A.M. - Verma P. - Chopra H. - Olea S.P. - Khan J. - Alvarez Suarez J.M. - Zheng X. - Tomczyk M. - Sabnani M.K. - Medina C.D.V. - Khalid G.M. - Boyina H.K. - Georgiev M.I. - Claudiu Supuran - Sobarzo-Sánchez E. - Fan T.P. - Pittala V. - Sureda A. - Braidy N. - Russo G.L. - Vacca R.A. - Banach M. - Lizard G. - Zarrouk A. - Hammami S. - Orhan I.E. - Aggarwal B.B. - Perry G. - Miller M.J. - Heinrich M. - Bishayee A. - Kijjoa A. - Arkells N. - Bredt D. - Wink M. - Fiebich B.l. - Kiran G. - Yeung A.W.K. - Gupta G.K. - Santini A. - Lucarini M. - Durazzo A. - El-Demerdash A. - Dinkova-Kostova A.T. - Cifuentes A. - Souto E.B. - Zubair M.A.M. - Badhe P. - Echeverría J. - Horbańczuk J.O. - Horbanczuk O.K. - Sheridan H. - Sheshe S.M. - Witkowska A.M. - Abu-Reidah I.M. - Riaz M. - Ullah H. - Oladipupo A.R. - Lopez V. - Sethiya N.K. - Shrestha B.G. - Ravanan P. - Gupta S.C.
Phytomedicine

4-Cyanamidobenzenesulfonamide derivatives: a novel class of human and bacterial carbonic anhydrase inhibitors

- Abdoli M. - Bonardi A. - Claudiu Supuran - Žalubovskis R.
Journal of Enzyme Inhibition and Medicinal Chemistry

2022

New β-arylchalcogeno amines with procognitive properties targeting Carbonic Anhydrases and Monoamine Oxidases

- Provensi G. - Costa A. - Rani B. - Becagli M.V. - Vaiano F. - Passani M.B. - Tanini D. - Capperucci A. - Carradori S. - Petzer J.P. - Petzer A. - Daniela Vullo - Costantino G. - Blandina P. - Angeli A. - Claudiu Supuran
European journal of medicinal chemistry

Carbonic Anhydrase Inhibition Activities of Schiff’s Bases Based on Quinazoline-Linked Benzenesulfonamide

- El-Azab A.S. - Abdel-Aziz A.A.M. - Ghabbour H.A. - Bua S. - Alessio Nocentini - Alkahtani H.M. - Alsaif N.A. - Al-Agamy M.H.M. - Claudiu Supuran
Molecules

New Dual P-Glycoprotein (P-gp) and Human Carbonic Anhydrase XII (hCA XII) Inhibitors as Multidrug Resistance (MDR) Reversers in Cancer Cells

- Braconi L. - Teodori E. - Riganti C. - Coronnello M. - Alessio Nocentini - Bartolucci G. - Pallecchi M. - Contino M. - Manetti D. - Romanelli M.N. - Claudiu Supuran - Dei S.
Journal of Medicinal Chemistry

Discovery of a Potent and Highly Selective Dipeptidyl Peptidase IV and Carbonic Anhydrase Inhibitor as “Antidiabesity” Agents Based on Repurposing and Morphing of WB-4101

- Artasensi A. - Angeli A. - Lammi C. - Bollati C. - Gervasoni S. - Baron G. - Matucci R. - Claudiu Supuran - Vistoli G. - Fumagalli L.
Journal of Medicinal Chemistry

Synthesis and anticancer activity of new benzensulfonamides incorporating s-triazines as cyclic linkers for inhibition of carbonic anhydrase IX

- Zain-Alabdeen A.I. - El-Moselhy T.F. - Sharafeldin N. - Angeli A. - Claudiu Supuran - El-Hamamsy M.H.
Scientific Reports

Dependence on linkers' flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents

- Tawfik H.O. - Belal A. - Abourehab M.A.S. - Angeli A. - Bonardi A. - Claudiu Supuran - El-Hamamsy M.H.
Journal of enzyme inhibition and medicinal chemistry

Development of benzene and benzothiazole-sulfonamide analogues as selective inhibitors of the tumor-associated carbonic anhydrase IX

- Manzoor S. - Angeli A. - Zara S. - Carradori S. - Rahman M.A. - Raza M.K. - Claudiu Supuran - Hoda N.
European Journal of Medicinal Chemistry

Carbonic Anhydrase inhibitors bearing organotelluride moieties as novel agents for antitumor therapy

- Petreni A. - Iacobescu A. - Simionescu N. - Petrovici A.R. - Angeli A. - Fifere A. - Pinteala M. - Claudiu Supuran
European Journal of Medicinal Chemistry

Design and synthesis of some new benzoylthioureido phenyl derivatives targeting carbonic anhydrase enzymes

- Najm M.A.A. - Mahmoud W.R. - Taher A.T. - Abbas S.E.S. - Awadallah F.M. - Allam H.A. - Daniela Vullo - Claudiu Supuran
Journal of Enzyme Inhibition and Medicinal Chemistry

Identification of New Carbonic Anhydrase VII Inhibitors by Structure-Based Virtual Screening

- Gantner M.E. - Prada Gori D.N. - Llanos M.A. - Talevi A. - Angeli A. - Daniela Vullo - Claudiu Supuran - Gavernet L.
Journal of Chemical Information and Modeling

Lipoyl-Based Antagonists of Transient Receptor Potential Cation A (TRPA1) Downregulate Osteosarcoma Cell Migration and Expression of Pro-Inflammatory Cytokines

- Francesconi O. - Corzana F. - Kontogianni G.I. - Pesciullesi G. - Gualdani R. - Claudiu Supuran - Angeli A. - Kavasi R.M. - Chatzinikolaidou M. - Nativi C.
ACS Pharmacology and Translational Science

Design and synthesis of benzothiazole-based SLC-0111 analogues as new inhibitors for the cancer-associated carbonic anhydrase isoforms IX and XII

- Al-Warhi T. - Elbadawi M.M. - Bonardi A. - Alessio Nocentini - Al-Karmalawy A.A. - Aljaeed N. - Alotaibi O.J. - Abdel-Aziz H.A. - Claudiu Supuran - Eldehna W.M.
Journal of Enzyme Inhibition and Medicinal Chemistry

The roles of plasma accessible and cytosolic carbonic anhydrases in bicarbonate (HCO3) excretion in Pacific hagfish (Eptatretus stoutii)

- Giacomin M. - Drummond J.M. - Claudiu Supuran - Goss G.G.
Journal of Comparative Physiology B: Biochemical, Systemic, and Environmental Physiology

Synthesis and biological evaluation of coumarin-thiazole hybrids as selective carbonic anhydrase IX and XII inhibitors

- Thacker P.S. - Newaskar V. - Angeli A. - Sigalapalli D.K. - Goud N.S. - Chirra H. - Shaik A.B. - Arifuddin M. - Claudiu Supuran
Archiv der Pharmazie

Inhibition studies of the protozoan α-carbonic anhydrase from Trypanosoma cruzi with phenols

- Bonardi A. - Parkkila S. - Claudiu Supuran
Journal of enzyme inhibition and medicinal chemistry

Squaramide-Tethered Sulfonamides and Coumarins: Synthesis, Inhibition of Tumor-Associated CAs IX and XII and Docking Simulations

- Arrighi G. - Puerta A. - Petrini A. - Hicke F.J. - Alessio Nocentini - Fernandes M.X. - Padrón J.M. - Claudiu Supuran - Fernández-Bolaños J.G. - López Ó.
International Journal of Molecular Sciences

Seleno Containing Compounds as Potent and Selective Antifungal Agents

- Angeli A. - Velluzzi A. - Selleri S. - Clemente Capasso - Spadini C. - Iannarelli M. - Cabassi C.S. - Fabrizio Carta - Claudiu Supuran
ACS Infectious Diseases

Discovery of novel drugs for Chagas disease: is carbonic anhydrase a target for antiprotozoal drugs?

- Beatriz Vermelho A. - Rodrigues G.C. - Alessio Nocentini - Mansoldo F.R.P. - Claudiu Supuran
Expert Opinion on Drug Discovery

Biochemical, structural, and computational studies of a γ-carbonic anhydrase from the pathogenic bacterium Burkholderia pseudomallei

- Di Fiore A. - De Luca V. - Langella E. - Alessio Nocentini - Buonanno M. - Monti S.M. - Claudiu Supuran - Clemente Capasso - De Simone G.
Computational and Structural Biotechnology Journal

Enaminone-based carboxylic acids as novel non-classical carbonic anhydrases inhibitors: design, synthesis and in vitro biological assessment

- Abo-Ashour M.F. - Almahli H. - Bonardia A. - Khalil A. - Al-Warhi T. - Al-Rashood S.T. - Abdel-Aziz H.A. - Alessio Nocentini - Claudiu Supuran - Eldehna W.M.
Journal of enzyme inhibition and medicinal chemistry

mGluR5 PAMs rescue cortical and behavioural defects in a mouse model of CDKL5 deficiency disorder

- Gurgone A. - Pizzo R. - Raspanti A. - Chiantia G. - Devi S. - Comai D. - Morello N. - Pilotto F. - Gnavi S. - Lupori L. - Mazziotti R. - Sagona G. - Putignano E. - Alessio Nocentini - Claudiu Supuran - Marcantoni A. - Pizzorusso T. - Giustetto M.
Neuropsychopharmacology

Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies

- Pontecorvi V. - Mori M. - Picarazzi F. - Zara S. - Carradori S. - Cataldi A. - Angeli A. - Berrino E. - Chimenti P. - Ciogli A. - Secci D. - Guglielmi P. - Claudiu Supuran
International journal of molecular sciences

Biochemical and Biophysical Characterization of Carbonic Anhydrase VI from Human Milk and Saliva

- Yrjänäinen A. - Patrikainen M.S. - Azizi L. - Tolvanen M.E.E. - Laitaoja M. - Jänis J. - Hytönen V.P. - Alessio Nocentini - Claudiu Supuran - Parkkila S.
Protein Journal

Preface

- Claudiu Supuran
Anti-Inflammatory and Anti-Allergy Agents in Medicinal Chemistry

Sulfonamide diuretic azosemide as an efficient carbonic anhydrase inhibitor

- Ferraroni M. - Angeli A. - Pinteala M. - Claudiu Supuran
Journal of Molecular Structure

Selective inhibition of carbonic anhydrase IX by sulphonylated 1,2,3-triazole incorporated benzenesulphonamides capable of inducing apoptosis

- Siwach K. - Kumar A. - Panchal H. - Kumar R. - Bhardwaj J.K. - Angeli A. - Claudiu Supuran - Sharma P.K.
Journal of Enzyme Inhibition and Medicinal Chemistry

Cloning, purification, kinetic and anion inhibition studies of a recombinant β-carbonic anhydrase from the Atlantic salmon parasite platyhelminth Gyrodactylus salaris

- Aspatwar A. - Barker H. - Aisala H. - Zueva K. - Kuuslahti M. - Tolvanen M. - Primmer C.R. - Lumme J. - Bonardi A. - Tripathi A. - Parkkila S. - Claudiu Supuran
Journal of Enzyme Inhibition and Medicinal Chemistry

4-(3-Alkyl/benzyl-guanidino)benzenesulfonamides as selective carbonic anhydrase VII inhibitors

- Abdoli M. - Giovannuzzi S. - Claudiu Supuran - Žalubovskis R.
Journal of Enzyme Inhibition and Medicinal Chemistry

Beta-Carbonic Anhydrase 1 from Trichomonas Vaginalis as New Antiprotozoan Drug Target

- Claudiu Supuran - Di Fiore A. - Parkkila S. - De Simone G.
Topics in Medicinal Chemistry

Correction to: Chagas Disease: Drug Development and Parasite Targets

- Vermelho A.B. - Cardoso V. - Mansoldo F.R.P. - Claudiu Supuran - Cedrola S.M.L. - Rodrigues I.A. - Rodrigues G.C.
Topics in Medicinal Chemistry

Chagas Disease: Drug Development and Parasite Targets

- Vermelho A.B. - Cardoso V. - Mansoldo F.R.P. - Claudiu Supuran - Cedrola S.M.L. - Rodrigues I.A. - Rodrigues G.C.
Topics in Medicinal Chemistry