Consorzio Interuniversitario per lo sviluppo dei Sistemi a Grande Interfase
Center for Colloid and Surface Science

PUBLICATIONS

Here you can find the updated list of all the publications of CSGI members and affilated staff. Please note that the only publications listed here are those published after the affilation of each member. If you are interested in the whole bibliography of CSGI members, including articles and books published before affilation to CSGI, please refer to academic research databases, such as Scopus, Web Of Science, Google Scholar, ect.

You can use the search bar below to filter the publication list.

2023

New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors

- Combs J. - Murat Bozdag - Cravey L.D. - Kota A. - McKenna R. - Angeli A. - Carta F. - Supuran C.T.
Molecules

2022

Small Molecule Alkoxy Oriented Selectiveness on Human Carbonic Anhydrase II and IX Inhibition

- Murat Bozdag - Cravey L. - Combs J. - Kota A. - McKenna R. - Angeli A. - Selleri S. - Carta F. - Supuran C.T.
ChemMedChem

New 1H-indole-2,3-dione 3-thiosemicarbazones with 3-sulfamoylphenyl moiety as selective carbonic anhydrase inhibitors

- Eraslan-Elma P. - Akdemir A. - Berrino E. - Murat Bozdag - Supuran C.T. - Karalı N.
Archiv der Pharmazie

2021

Privileged scaffolds in medicinal chemistry: Studies on pyrazolo[1,5-a]pyrimidines on sulfonamide containing Carbonic Anhydrase inhibitors

- Gumus A. - Murat Bozdag - Angeli A. - Peat T.S. - Carta F. - Supuran C.T. - Selleri S.
Bioorganic and Medicinal Chemistry Letters

2020

In vitro inhibition of Mycobacterium tuberculosis β-carbonic anhydrase 3 with Mono- and dithiocarbamates and evaluation of their toxicity using zebrafish developing embryos

- Aspatwar A. - Hammaren M. - Parikka M. - Parkkila S. - Carta F. - Murat Bozdag - Daniela Vullo - Supuran C.
Journal of Enzyme Inhibition and Medicinal Chemistry

Benzylaminoethyureido-tailed benzenesulfonamides: Design, synthesis, kinetic and X-ray investigations on human carbonic anhydrases

- Ali M. - Murat Bozdag - Farooq U. - Angeli A. - Carta F. - Berto P. - Zanotti G. - Supuran C.T.
International Journal of Molecular Sciences

Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors

- Berrino E. - Angeli A. - Zhdanov D.D. - Kiryukhina A.P. - Milaneschi A. - De Luca A. - Murat Bozdag - Carradori S. - Selleri S. - Bartolucci G. - Peat T.S. - Ferraroni M. - Supuran C.T. - Carta F.
Journal of Medicinal Chemistry

2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site

- Murat Bozdag - Supuran C.T. - Esposito D. - Angeli A. - Carta F. - Monti S.M. - De Simone G. - Alterio V.
Chemical Communications

"a Sweet Combination": Developing Saccharin and Acesulfame K Structures for Selectively Targeting the Tumor-Associated Carbonic Anhydrases IX and XII

- Bua S. - Lomelino C. - Murray A.B. - Osman S.M. - Alothman Z.A. - Murat Bozdag - Abdel-Aziz H.A. - Eldehna W.M. - McKenna R. - Nocentini A. - Supuran C.T.
Journal of Medicinal Chemistry

2019

State of the art on carbonic anhydrase modulators for biomedical purposes

- Murat Bozdag - Altamimi A.S.A. - Daniela Vullo - Supuran C.T. - Carta F.
Current Medicinal Chemistry

Pain relieving effect of-NSAIDS-CAIs hybrid molecules: Systemic and intra-articular treatments against rheumatoid arthritis

- Micheli L. - Murat Bozdag - Akgul O. - Carta F. - Guccione C. - Bergonzi M. - Anna Rita Bilia - Cinci L. - Lucarini E. - Parisio C. - Supuran C. - Ghelardini C. - Di Cesare Mannelli L.
International Journal of Molecular Sciences

A non-catalytic function of carbonic anhydrase IX contributes to the glycolytic phenotype and pH regulation in human breast cancer cells

- Mboge M. - Chen Z. - Khokhar D. - Wolff A. - Ai L. - Heldermon C. - Murat Bozdag - Carta F. - Supuran C. - Brown K. - McKenna R. - Frost C. - Frost S.
Biochemical Journal

N-aryl-N’-ureido-O-sulfamates: Potent and selective inhibitors of the human Carbonic Anhydrase VII isoform with neuropathic pain relieving properties

- Murat Bozdag - Poli G. - Angeli A. - Lucarini E. - Tuccinardi T. - Di Cesare Mannelli L. - Selleri S. - Ghelardini C. - Winum J.Y. - Carta F. - Supuran C.T.
Bioorganic Chemistry

Synthesis and evaluation of carbonic anhydrase inhibitors with carbon monoxide releasing properties for the management of rheumatoid arthritis

- Berrino E. - Milazzo L. - Micheli L. - Daniela Vullo - Angeli A. - Murat Bozdag - Nocentini A. - Menicatti M. - Bartolucci G. - Di Cesare Mannelli L. - Ghelardini C. - Supuran C.T. - Carta F.
Journal of Medicinal Chemistry

Mycobacterium tuberculosis β-carbonic anhydrases: Novel targets for developing antituberculosis drugs

- Aspatwar A. - Kairys V. - Rala S. - Parikka M. - Murat Bozdag - Carta F. - Supuran C.T. - Parkkila S.
International Journal of Molecular Sciences

Carbonic anhydrase inhibitors based on sorafenib scaffold: Design, synthesis, crystallographic investigation and effects on primary breast cancer cells

- Murat Bozdag - Ferraroni M. - Ward C. - Carta F. - Bua S. - Angeli A. - Langdon S.P. - Kunkler I.H. - Al-Tamimi A.M.S. - Supuran C.T.
European Journal of Medicinal Chemistry

Mechanisms of action of carbonic anhydrase inhibitors: Compounds that anchor to the zinc-bound nucleophile

- Murat Bozdag - Angeli A. - Tanc M.
Carbonic Anhydrases: Biochemistry and Pharmacology of an Evergreen Pharmaceutical Target

2018

Mono- and di-thiocarbamate inhibition studies of the δ-carbonic anhydrase TweCAδ from the marine diatom Thalassiosira weissflogii

- Bua S. - Murat Bozdag - Del Prete S. - Carta F. - Donald W. - Clemente Capasso - Supuran C.
Journal of Enzyme Inhibition and Medicinal Chemistry

Discovery of 4-Hydroxy-3-(3-(phenylureido)benzenesulfonamides as SLC-0111 Analogues for the Treatment of Hypoxic Tumors Overexpressing Carbonic Anhydrase IX

- Murat Bozdag - Carta F. - Ceruso M. - Ferraroni M. - McDonald P.C. - Dedhar S. - Supuran C.T.
Journal of Medicinal Chemistry

Synthesis of N′-phenyl-N-hydroxyureas and investigation of their inhibitory activities on human carbonic anhydrases

- Murat Bozdag - Carta F. - Angeli A. - Osman S. - Alasmary F. - AlOthman Z. - Supuran C.
Bioorganic Chemistry

Selective inhibition of carbonic anhydrase IX over carbonic anhydrase XII in breast cancer cells using benzene sulfonamides: Disconnect between activity and growth inhibition

- Mboge M.Y. - Chen Z. - Wolff A. - Mathias J.V. - Tu C. - Brown K.D. - Murat Bozdag - Carta F. - Supuran C.T. - McKenna R. - Frost S.C.
PLoS ONE

Inhibition of α-, β-, γ-, and δ-carbonic anhydrases from bacteria and diatoms with N′-aryl-N-hydroxy-ureas

- Berrino E. - Murat Bozdag - Del Prete S. - Alasmary F. - Alqahtani L. - AlOthman Z. - Clemente Capasso - Supuran C.
Journal of Enzyme Inhibition and Medicinal Chemistry

Inhibition of carbonic anhydrases by a substrate analog: benzyl carbamate directly coordinates the catalytic zinc ion mimicking bicarbonate binding

- De Simone G. - Angeli A. - Murat Bozdag - Supuran C.T. - Winum J.Y. - Monti S.M. - Alterio V.
Chemical Communications

2017

Carbonic anhydrase I, II, IV and IX inhibition with a series of 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives

- Murat Bozdag - Bua S. - Osman S. - AlOthman Z. - Supuran C.
Journal of Enzyme Inhibition and Medicinal Chemistry

Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides

- Abdoli M. - Angeli A. - Murat Bozdag - Carta F. - Kakanejadifard A. - Saeidian H. - Supuran C.
Journal of Enzyme Inhibition and Medicinal Chemistry

Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa

- Daniela Vullo - Del Prete S. - Nocentini A. - Osman S. - AlOthman Z. - Clemente Capasso - Murat Bozdag - Carta F. - Gratteri P. - Supuran C.
Bioorganic and Medicinal Chemistry

2016

Synthesis 4-[2-(2-mercapto-4-oxo-4H-quinazolin-3-yl)-ethyl]-benzenesulfonamides with subnanomolar carbonic anhydrase II and XII inhibitory properties

- Murat Bozdag - Alafeefy A. - Carta F. - Ceruso M. - Al-Tamimi A. - Al-Kahtani A. - Alasmary F. - Supuran C.
Bioorganic and Medicinal Chemistry

Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase

- Murat Bozdag - Carta F. - Daniela Vullo - Isik S. - AlOthman Z. - Osman S.M. - Andrea Scozzafava - Supuran C.T.
Journal of Enzyme Inhibition and Medicinal Chemistry

2015

Synthesis of a novel affinity gel for the purification of carbonic anhydrases

- Murat Bozdag - Isik S. - Beyaztas S. - Arslan O. - Supuran C.
Journal of Enzyme Inhibition and Medicinal Chemistry

Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity

- Murat Bozdag - Alafeefy A.M. - Daniela Vullo - Carta F. - Dedeoglu N. - Al-Tamimi A.M.S. - Al-Jaber N.A. - Andrea Scozzafava - Supuran C.T.
Bioorganic and Medicinal Chemistry

2014

Next-generation dithiocarbamate carbonic anhydrase inhibitors

- Carta F. - Murat Bozdag - Tanc M. - Supuran C.
Targeting Carbonic Anhydrases

Structural insights on carbonic anhydrase inhibitory action, isoform selectivity, and potency of sulfonamides and coumarins incorporating arylsulfonylureido groups

- Murat Bozdag - Ferraroni M. - Carta F. - Daniela Vullo - Lucarini L. - Orlandini E. - Rossello A. - Nuti E. - Andrea Scozzafava - Masini E. - Supuran C.
Journal of Medicinal Chemistry

2013

Novel small molecule protein arginine deiminase 4 (PAD4) inhibitors

- Murat Bozdag - Dreker T. - Henry C. - Tosco P. - Vallaro M. - Fruttero R. - Andrea Scozzafava - Carta F. - Supuran C.T.
Bioorganic and Medicinal Chemistry Letters