Here you can find the updated list of all the publications of CSGI members and affilated staff. Please note that the only publications listed here are those published after the affilation of each member. If you are interested in the whole bibliography of CSGI members, including articles and books published before affilation to CSGI, please refer to academic research databases, such as Scopus, Web Of Science, Google Scholar, ect.
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Production, crystallographic studies, and functional profiling of γ-carbonic anhydrase from the probiotic Limosilactobacillus reuteri: In vitro and cell-based insights
- Bonardi A. - Carradori S. - Paoletti N. - Andrea Angeli - Ferraroni M. - Iacovozzi D. - Gallorini M. - D'Agostino I. - De Luca V. - Gratteri P. - Cataldi A. - Supuran C.T. - Clemente CapassoDiscovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells
- Murat Bozdag - Mroweh N. - Raucci A. - Andrea Angeli - Peppicelli S. - Biagioni A. - Calorini L. - Trisciuoglio D. - Ragno R. - Astolfi R. - Giuliani L. - Zwergel C. - Valente S. - Andreucci E. - Carta F. - Mai A. - Supuran C.T.Coumarin-Containing Aromatic Sulfonamides With Carbonic Anhydrase Inhibitory Properties Against Human and Fungal Isoforms
- Andrea Angeli - Petrou A. - Kartsev V. - De Luca V. - Clemente Capasso - Geronikaki A. - Supuran C.T.Design and Synthesis of Ketoconazole Derivatives as Innovative Anti-Infective Agents
- Renzi G. - Andrea Angeli - Selleri S. - Spadini C. - Mezzasalma N. - Hull M.T. - Kelly S.L. - Clemente Capasso - Cabassi C.S. - Carta F. - Supuran C.T.Pegylation approach applied to erlotinib-carbonic anhydrase inhibitors hybrids towards anticancer agents
- Filiberti S. - Renzi G. - Carta F. - Fantacuzzi M. - D'Agostino I. - Benito G. - Andrea Angeli - Massardi M.L. - Simsek R. - Clemente Capasso - Carradori S. - Ronca R. - Supuran C.T.Hitting Two Birds With One Stone: Dual Modulation of Brain Carbonic Anhydrases and Histone Deacetylases Boosts Memory Consolidation
- Costa A. - Murat Bozdag - Renzi G. - Rani B. - Passani M.B. - Andrea Angeli - Provensi G. - Carta F. - Supuran C.T.A Journey Around Boronic Acids: Sulfonyl Hydrazone-Containing Derivatives as Carbonic Anhydrase Inhibitors
- Anakök D.A. - Andrea Angeli - D'Agostino I. - Renzi G. - Massardi M.L. - Tavani C. - Çete S. - Carradori S. - Ronca R. - Clemente Capasso - Carta F. - Supuran C.T.O-derivatization of natural tropolone and β-thujaplicin leading to effective inhibitors of human carbonic anhydrases IX and XII
- Melfi F. - D'Agostino I. - Carradori S. - Carta F. - Andrea Angeli - Costa G. - Renzi G. - Čikoš A. - Daniela Vullo - Rešetar J. - Ferraroni M. - Baroni C. - Mancuso F. - Gitto R. - Ambrosio F.A. - Marchese E. - Torcasio R. - Amodio N. - Clemente Capasso - Alcaro S. - Supuran C.T. Structural Studies of the Dopamine D
Kinetic and structural studies of gamma-carbonic anhydrase from the oral pathogen Porphyromonas gingivalis
- Ferraroni M. - Andrea Angeli - De Luca V. - Clemente Capasso - Supuran C.T.Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study
- Marinacci B. - D’Agostino I. - Andrea Angeli - Carradori S. - Melfi F. - Grande R. - Corsiani M. - Ferraroni M. - Agamennone M. - Tondo A.R. - Zara S. - Puca V. - Pellegrini B. - Vagaggini C. - Dreassi E. - Patrauchan M.A. - Clemente Capasso - Nicolotti O. - Carta F. - Supuran C.T. Phosphorylation strongly affects the inhibition of human carbonic anhydrase I CO
Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α-carbonic anhydrase inhibitors
- Gumus A. - D'Agostino I. - Puca V. - Crocetta V. - Carradori S. - Cutarella L. - Mori M. - Carta F. - Andrea Angeli - Clemente Capasso - Supuran C.T.Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori: Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies
- Giampietro L. - Marinacci B. - Della Valle A. - D’Agostino I. - Lauro A. - Mori M. - Carradori S. - Ammazzalorso A. - De Filippis B. - Maccallini C. - Andrea Angeli - Clemente Capasso - Francati S. - Mollica A. - Grande R. - Supuran C.T. Comparative CO
Direct assembly of N-sulfamoyl lactam scaffolds bearing a zinc-binding group for inhibiting metalloenzymes based on desymmetrization of sulfamide and the Castagnoli-Cushman reaction
- Karchuganova E. - Martynova S. - Kalinin S. - Andrea Angeli - Dar'in D. - Daniela Vullo - Supuran C.T. - Bakulina O. The dopamine D
Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based Inhibitors
- De Luca V. - Andrea Angeli - Nocentini Alessio - Gratteri P. - Pratesi S. - Tanini D. - Carginale V. - Capperucci A. - Supuran C.T. - Clemente CapassoNovel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy
- Andrea Angeli - Chelli I. - Lucarini L. - Sgambellone S. - Marri S. - Villano S. - Ferraroni M. - De Luca V. - Clemente Capasso - Carta F. - Supuran C.T.Antimalarial Agents Targeting Plasmodium falciparum Carbonic Anhydrase: Towards Artesunate Hybrid Compounds with Dual Mechanism of Action
- D'Agostino I. - Zara S. - Carradori S. - De Luca V. - Clemente Capasso - Kocken C.H.M. - Zeeman A.M. - Andrea Angeli - Carta F. - Supuran C.T.Photoactivatable Heptamethine-Based Carbonic Anhydrase Inhibitors Leading to New Anti-Antibacterial Agents
- Carradori S. - Andrea Angeli - Sfragano P.S. - Yzeiri X. - Calamante M. - Tanini D. - Capperucci A. - Kunstek H. - Varbanov M. - Clemente Capasso - Supuran C.T.Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships
- Fantacuzzi M. - D’Agostino I. - Carradori S. - Liguori F. - Carta F. - Agamennone M. - Andrea Angeli - Sannio F. - Docquier J.D. - Clemente Capasso - Supuran C.T.New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors
- Combs J. - Murat Bozdag - Cravey L.D. - Kota A. - McKenna R. - Andrea Angeli - Carta F. - Supuran C.T.Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors
- Andrea Angeli - Petrou A. - Kartsev V. - Lichitsky B. - Komogortsev A. - Clemente Capasso - Geronikaki A. - Supuran C.T.One-Pot Procedure for the Synthesis of Asymmetric Substituted Ureido Benzene Sulfonamides as Effective Inhibitors of Carbonic Anhydrase Enzymes
- Vannozzi G. - Daniela Vullo - Andrea Angeli - Ferraroni M. - Combs J. - Lomelino C. - Andring J. - McKenna R. - Bartolucci G. - Pallecchi M. - Lucarini L. - Sgambellone S. - Masini E. - Carta F. - Supuran C.T.Heterologous expression and biochemical characterisation of the recombinant β-carbonic anhydrase (MpaCA) from the warm-blooded vertebrate pathogen malassezia pachydermatis
- De Luca V. - Andrea Angeli - Mazzone V. - Adelfio C. - Carginale V. - Scaloni A. - Carta F. - Selleri S. - Supuran C.T. - Clemente CapassoSeleno Containing Compounds as Potent and Selective Antifungal Agents
- Andrea Angeli - Velluzzi A. - Selleri S. - Clemente Capasso - Spadini C. - Iannarelli M. - Cabassi C.S. - Carta F. - Supuran C.T.Small Molecule Alkoxy Oriented Selectiveness on Human Carbonic Anhydrase II and IX Inhibition
- Murat Bozdag - Cravey L. - Combs J. - Kota A. - McKenna R. - Andrea Angeli - Selleri S. - Carta F. - Supuran C.T.Thiosemicarbazide-Substituted Coumarins as Selective Inhibitors of the Tumor Associated Human Carbonic Anhydrases IX and XII
- Gumus A. - Murat Bozdag - Akdemir A. - Andrea Angeli - Selleri S. - Carta F. - Supuran C.T.New β-arylchalcogeno amines with procognitive properties targeting Carbonic Anhydrases and Monoamine Oxidases
- Provensi G. - Costa A. - Rani B. - Becagli M.V. - Vaiano F. - Passani M.B. - Tanini D. - Capperucci A. - Carradori S. - Petzer J.P. - Petzer A. - Daniela Vullo - Costantino G. - Blandina P. - Andrea Angeli - Supuran C.T.Activation studies with amino acids and amines of a β-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri previously annotated as Staphylococcus aureus (SauBCA) carbonic anhydrase
- Andrea Angeli - Urbański L.J. - Clemente Capasso - Parkkila S. - Supuran C.T.Identification of New Carbonic Anhydrase VII Inhibitors by Structure-Based Virtual Screening
- Gantner M.E. - Prada Gori D.N. - Llanos M.A. - Talevi A. - Andrea Angeli - Daniela Vullo - Supuran C.T. - Gavernet L.Synthesis and biological evaluation of sulfonamide-based compounds as inhibitors of carbonic anhydrase from Vibrio cholerae
- Mancuso F. - Andrea Angeli - De Luca V. - Bucolo F. - De Luca L. - Clemente Capasso - Supuran C.T. - Gitto R.Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase
- Nocentini Alessio - Andrea Angeli - Carta F. - Winum J.Y. - Zalubovskis R. - Carradori S. - Clemente Capasso - Donald W.A. - Supuran C.T.Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors
- Andrea Angeli - Carta F. - Nocentini Alessio - Winum J.Y. - Zalubovskis R. - Onnis V. - Eldehna W.M. - Clemente Capasso - Carradori S. - Donald W.A. - Dedhar S. - Supuran C.T.Taurultams incorporating arylsulfonamide: First in vitro inhibition studies of α-, β- and γ-class Carbonic Anhydrases from Vibrio cholerae and Burkholderia pseudomallei
- Akgul O. - Andrea Angeli - Selleri S. - Clemente Capasso - Supuran C.T. - Carta F.Inhibitory effects of sulfonamide derivatives on the β‐carbonic anhydrase (Mpaca) from malassezia pachydermatis, a commensal, pathogenic fungus present in domestic animals
- De Luca V. - Andrea Angeli - Mazzone V. - Adelfio C. - Carta F. - Selleri S. - Carginale V. - Scaloni A. - Supuran C.T. - Clemente CapassoPrivileged scaffolds in medicinal chemistry: Studies on pyrazolo[1,5-a]pyrimidines on sulfonamide containing Carbonic Anhydrase inhibitors
- Gumus A. - Murat Bozdag - Andrea Angeli - Peat T.S. - Carta F. - Supuran C.T. - Selleri S.Glyco-Coated CdSe/ZnS Quantum Dots as Nanoprobes for Carbonic Anhydrase IX Imaging in Cancer Cells
- Giacomo Biagiotti - Andrea Angeli - Giacomini A. - Toniolo G. - Landini L. - Salerno G. - Di Cesare Mannelli L. - Ghelardini C. - Mello T. - Mussi S. - Ravelli C. - Marelli M. - Cicchi S. - Menna E. - Ronca R. - Supuran C.T. - Barbara Richichi4-Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae
- Mancuso F. - De Luca L. - Bucolo F. - Vrabel M. - Andrea Angeli - Clemente Capasso - Supuran C.T. - Gitto R.New sulfanilamide derivatives incorporating heterocyclic carboxamide moieties as carbonic anhydrase inhibitors
- Andrea Angeli - Kartsev V. - Petrou A. - Pinteala M. - Vydzhak R.M. - Panchishin S.Y. - Brovarets V. - De Luca V. - Clemente Capasso - Geronikaki A. - Supuran C.T.Selective inhibition of helicobacter pylori carbonic anhydrases by carvacrol and thymol could impair biofilm production and the release of outer membrane vesicles
- Grande R. - Carradori S. - Puca V. - Vitale I. - Andrea Angeli - Nocentini Alessio - Bonardi A. - Gratteri P. - Lanuti P. - Bologna G. - Simeone P. - Clemente Capasso - De Luca V. - Supuran C.T.Phenols from Origanum dictamnus L. and Thymus vulgaris L. and their activity against Malassezia globosa carbonic anhydrase
- Paloukopoulou C. - Govari S. - Soulioti A. - Stefanis I. - Andrea Angeli - Matheeussen A. - Clemente Capasso - Cos P. - Supuran C.T. - Karioti A.Design, synthesis, and biological evaluation of selective hCA IX inhibitors
- Carta F. - Daniela Vullo - Andrea AngeliUnconventional amino acids in medicinal chemistry: First report on taurine merged within carbonic anhydrase inhibitors
- Akgül Ö. - Andrea Angeli - Daniela Vullo - Carta F. - Supuran C.T.Evaluation of thio-and seleno-acetamides bearing benzenesulfonamide as inhibitor of carbonic anhydrases from different pathogenic bacteria
- Andrea Angeli - Pinteala M. - Maier S.S. - Simionescu B.C. - Milaneschi A. - Abbas G. - Del Prete S. - Clemente Capasso - Capperucci A. - Tanini D. - Carta F. - Supuran C.T.Crystal structure of a tetrameric type II β-carbonic anhydrase from the pathogenic bacterium burkholderia pseudomallei
- Andrea Angeli - Ferraroni M. - Pinteala M. - Maier S.S. - Simionescu B.C. - Carta F. - Del Prete S. - Clemente Capasso - Supuran C.T.Carbonic anhydrase inhibitors targeting metabolism and tumor microenvironment
- Andrea Angeli - Carta F. - Nocentini Alessio - Winum J.Y. - Zalubovskis R. - Akdemir A. - Onnis V. - Eldehna W.M. - Clemente Capasso - Simone G.D. - Monti S.M. - Carradori S. - Donald W.A. - Dedhar S. - Supuran C.T.Benzylaminoethyureido-tailed benzenesulfonamides: Design, synthesis, kinetic and X-ray investigations on human carbonic anhydrases
- Ali M. - Murat Bozdag - Farooq U. - Andrea Angeli - Carta F. - Berto P. - Zanotti G. - Supuran C.T.N-aryl-N′-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: Deciphering the binding mode of new potential agents in mitochondrial dysfunctions
- Poli G. - Murat Bozdag - Berrino E. - Andrea Angeli - Tuccinardi T. - Carta F. - Supuran C.T.