Consorzio Interuniversitario per lo sviluppo dei Sistemi a Grande Interfase
Center for Colloid and Surface Science

PUBLICATIONS

Here you can find the updated list of all the publications of CSGI members and affilated staff. Please note that the only publications listed here are those published after the affilation of each member. If you are interested in the whole bibliography of CSGI members, including articles and books published before affilation to CSGI, please refer to academic research databases, such as Scopus, Web Of Science, Google Scholar, ect.

You can use the search bar below to filter the publication list.

2026

Production, crystallographic studies, and functional profiling of γ-carbonic anhydrase from the probiotic Limosilactobacillus reuteri: In vitro and cell-based insights

- Bonardi A. - Carradori S. - Paoletti N. - Andrea Angeli - Ferraroni M. - Iacovozzi D. - Gallorini M. - D'Agostino I. - De Luca V. - Gratteri P. - Cataldi A. - Supuran C.T. - Clemente Capasso
European Journal of Medicinal Chemistry

2025

Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells

- Murat Bozdag - Mroweh N. - Raucci A. - Andrea Angeli - Peppicelli S. - Biagioni A. - Calorini L. - Trisciuoglio D. - Ragno R. - Astolfi R. - Giuliani L. - Zwergel C. - Valente S. - Andreucci E. - Carta F. - Mai A. - Supuran C.T.
Journal of Medicinal Chemistry

Coumarin-Containing Aromatic Sulfonamides With Carbonic Anhydrase Inhibitory Properties Against Human and Fungal Isoforms

- Andrea Angeli - Petrou A. - Kartsev V. - De Luca V. - Clemente Capasso - Geronikaki A. - Supuran C.T.
Chemical Biology and Drug Design

Design and Synthesis of Ketoconazole Derivatives as Innovative Anti-Infective Agents

- Renzi G. - Andrea Angeli - Selleri S. - Spadini C. - Mezzasalma N. - Hull M.T. - Kelly S.L. - Clemente Capasso - Cabassi C.S. - Carta F. - Supuran C.T.
Archiv Der Pharmazie

Pegylation approach applied to erlotinib-carbonic anhydrase inhibitors hybrids towards anticancer agents

- Filiberti S. - Renzi G. - Carta F. - Fantacuzzi M. - D'Agostino I. - Benito G. - Andrea Angeli - Massardi M.L. - Simsek R. - Clemente Capasso - Carradori S. - Ronca R. - Supuran C.T.
Rsc Medicinal Chemistry

Hitting Two Birds With One Stone: Dual Modulation of Brain Carbonic Anhydrases and Histone Deacetylases Boosts Memory Consolidation

- Costa A. - Murat Bozdag - Renzi G. - Rani B. - Passani M.B. - Andrea Angeli - Provensi G. - Carta F. - Supuran C.T.
Archiv Der Pharmazie

A Journey Around Boronic Acids: Sulfonyl Hydrazone-Containing Derivatives as Carbonic Anhydrase Inhibitors

- Anakök D.A. - Andrea Angeli - D'Agostino I. - Renzi G. - Massardi M.L. - Tavani C. - Çete S. - Carradori S. - Ronca R. - Clemente Capasso - Carta F. - Supuran C.T.
Chemical Biology and Drug Design

O-derivatization of natural tropolone and β-thujaplicin leading to effective inhibitors of human carbonic anhydrases IX and XII

- Melfi F. - D'Agostino I. - Carradori S. - Carta F. - Andrea Angeli - Costa G. - Renzi G. - Čikoš A. - Daniela Vullo - Rešetar J. - Ferraroni M. - Baroni C. - Mancuso F. - Gitto R. - Ambrosio F.A. - Marchese E. - Torcasio R. - Amodio N. - Clemente Capasso - Alcaro S. - Supuran C.T.
European Journal of Medicinal Chemistry

2024

Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study

- Marinacci B. - D’Agostino I. - Andrea Angeli - Carradori S. - Melfi F. - Grande R. - Corsiani M. - Ferraroni M. - Agamennone M. - Tondo A.R. - Zara S. - Puca V. - Pellegrini B. - Vagaggini C. - Dreassi E. - Patrauchan M.A. - Clemente Capasso - Nicolotti O. - Carta F. - Supuran C.T.
Journal of Medicinal Chemistry

Phosphorylation strongly affects the inhibition of human carbonic anhydrase I CO2 hydration activity

- Andrea Angeli - De Luca V. - Huang X. - Winter D.L. - Clemente Capasso - Supuran C.T. - Donald W.A.
Archives of Biochemistry and Biophysics

Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α-carbonic anhydrase inhibitors

- Gumus A. - D'Agostino I. - Puca V. - Crocetta V. - Carradori S. - Cutarella L. - Mori M. - Carta F. - Andrea Angeli - Clemente Capasso - Supuran C.T.
Archiv der Pharmazie

Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori: Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies

- Giampietro L. - Marinacci B. - Della Valle A. - D’Agostino I. - Lauro A. - Mori M. - Carradori S. - Ammazzalorso A. - De Filippis B. - Maccallini C. - Andrea Angeli - Clemente Capasso - Francati S. - Mollica A. - Grande R. - Supuran C.T.
Pharmaceuticals

Comparative CO2 and SiO2 hydratase activity of an enzyme from the siliceous demosponge Suberites domuncula

- Andrea Angeli - De Luca V. - Clemente Capasso - Di Costanzo L.F. - Supuran C.T.
Archives of Biochemistry and Biophysics

Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based Inhibitors

- De Luca V. - Andrea Angeli - Nocentini Alessio - Gratteri P. - Pratesi S. - Tanini D. - Carginale V. - Capperucci A. - Supuran C.T. - Clemente Capasso
International journal of molecular sciences

2023

Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy

- Andrea Angeli - Chelli I. - Lucarini L. - Sgambellone S. - Marri S. - Villano S. - Ferraroni M. - De Luca V. - Clemente Capasso - Carta F. - Supuran C.T.
Journal of Medicinal Chemistry

Antimalarial Agents Targeting Plasmodium falciparum Carbonic Anhydrase: Towards Artesunate Hybrid Compounds with Dual Mechanism of Action

- D'Agostino I. - Zara S. - Carradori S. - De Luca V. - Clemente Capasso - Kocken C.H.M. - Zeeman A.M. - Andrea Angeli - Carta F. - Supuran C.T.
ChemMedChem

Photoactivatable Heptamethine-Based Carbonic Anhydrase Inhibitors Leading to New Anti-Antibacterial Agents

- Carradori S. - Andrea Angeli - Sfragano P.S. - Yzeiri X. - Calamante M. - Tanini D. - Capperucci A. - Kunstek H. - Varbanov M. - Clemente Capasso - Supuran C.T.
International Journal of Molecular Sciences

Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships

- Fantacuzzi M. - D’Agostino I. - Carradori S. - Liguori F. - Carta F. - Agamennone M. - Andrea Angeli - Sannio F. - Docquier J.D. - Clemente Capasso - Supuran C.T.
Journal of Enzyme Inhibition and Medicinal Chemistry

New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors

- Combs J. - Murat Bozdag - Cravey L.D. - Kota A. - McKenna R. - Andrea Angeli - Carta F. - Supuran C.T.
Molecules

Synthesis, Biological and In Silico Studies of Griseofulvin and Usnic Acid Sulfonamide Derivatives as Fungal, Bacterial and Human Carbonic Anhydrase Inhibitors

- Andrea Angeli - Petrou A. - Kartsev V. - Lichitsky B. - Komogortsev A. - Clemente Capasso - Geronikaki A. - Supuran C.T.
International Journal of Molecular Sciences

2022

One-Pot Procedure for the Synthesis of Asymmetric Substituted Ureido Benzene Sulfonamides as Effective Inhibitors of Carbonic Anhydrase Enzymes

- Vannozzi G. - Daniela Vullo - Andrea Angeli - Ferraroni M. - Combs J. - Lomelino C. - Andring J. - McKenna R. - Bartolucci G. - Pallecchi M. - Lucarini L. - Sgambellone S. - Masini E. - Carta F. - Supuran C.T.
Journal of Medicinal Chemistry

Heterologous expression and biochemical characterisation of the recombinant β-carbonic anhydrase (MpaCA) from the warm-blooded vertebrate pathogen malassezia pachydermatis

- De Luca V. - Andrea Angeli - Mazzone V. - Adelfio C. - Carginale V. - Scaloni A. - Carta F. - Selleri S. - Supuran C.T. - Clemente Capasso
Journal of Enzyme Inhibition and Medicinal Chemistry

Seleno Containing Compounds as Potent and Selective Antifungal Agents

- Andrea Angeli - Velluzzi A. - Selleri S. - Clemente Capasso - Spadini C. - Iannarelli M. - Cabassi C.S. - Carta F. - Supuran C.T.
ACS Infectious Diseases

Small Molecule Alkoxy Oriented Selectiveness on Human Carbonic Anhydrase II and IX Inhibition

- Murat Bozdag - Cravey L. - Combs J. - Kota A. - McKenna R. - Andrea Angeli - Selleri S. - Carta F. - Supuran C.T.
ChemMedChem

New β-arylchalcogeno amines with procognitive properties targeting Carbonic Anhydrases and Monoamine Oxidases

- Provensi G. - Costa A. - Rani B. - Becagli M.V. - Vaiano F. - Passani M.B. - Tanini D. - Capperucci A. - Carradori S. - Petzer J.P. - Petzer A. - Daniela Vullo - Costantino G. - Blandina P. - Andrea Angeli - Supuran C.T.
European journal of medicinal chemistry

Identification of New Carbonic Anhydrase VII Inhibitors by Structure-Based Virtual Screening

- Gantner M.E. - Prada Gori D.N. - Llanos M.A. - Talevi A. - Andrea Angeli - Daniela Vullo - Supuran C.T. - Gavernet L.
Journal of Chemical Information and Modeling

Synthesis and biological evaluation of sulfonamide-based compounds as inhibitors of carbonic anhydrase from Vibrio cholerae

- Mancuso F. - Andrea Angeli - De Luca V. - Bucolo F. - De Luca L. - Clemente Capasso - Supuran C.T. - Gitto R.
Archiv der Pharmazie

2021

Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase

- Nocentini Alessio - Andrea Angeli - Carta F. - Winum J.Y. - Zalubovskis R. - Carradori S. - Clemente Capasso - Donald W.A. - Supuran C.T.
Journal of Enzyme Inhibition and Medicinal Chemistry

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors

- Andrea Angeli - Carta F. - Nocentini Alessio - Winum J.Y. - Zalubovskis R. - Onnis V. - Eldehna W.M. - Clemente Capasso - Carradori S. - Donald W.A. - Dedhar S. - Supuran C.T.
Biophysical Journal

Inhibitory effects of sulfonamide derivatives on the β‐carbonic anhydrase (Mpaca) from malassezia pachydermatis, a commensal, pathogenic fungus present in domestic animals

- De Luca V. - Andrea Angeli - Mazzone V. - Adelfio C. - Carta F. - Selleri S. - Carginale V. - Scaloni A. - Supuran C.T. - Clemente Capasso
International Journal of Molecular Sciences

Privileged scaffolds in medicinal chemistry: Studies on pyrazolo[1,5-a]pyrimidines on sulfonamide containing Carbonic Anhydrase inhibitors

- Gumus A. - Murat Bozdag - Andrea Angeli - Peat T.S. - Carta F. - Supuran C.T. - Selleri S.
Bioorganic and Medicinal Chemistry Letters

Glyco-Coated CdSe/ZnS Quantum Dots as Nanoprobes for Carbonic Anhydrase IX Imaging in Cancer Cells

- Giacomo Biagiotti - Andrea Angeli - Giacomini A. - Toniolo G. - Landini L. - Salerno G. - Di Cesare Mannelli L. - Ghelardini C. - Mello T. - Mussi S. - Ravelli C. - Marelli M. - Cicchi S. - Menna E. - Ronca R. - Supuran C.T. - Barbara Richichi
ACS Applied Nano Materials

4-Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae

- Mancuso F. - De Luca L. - Bucolo F. - Vrabel M. - Andrea Angeli - Clemente Capasso - Supuran C.T. - Gitto R.
ChemMedChem

New sulfanilamide derivatives incorporating heterocyclic carboxamide moieties as carbonic anhydrase inhibitors

- Andrea Angeli - Kartsev V. - Petrou A. - Pinteala M. - Vydzhak R.M. - Panchishin S.Y. - Brovarets V. - De Luca V. - Clemente Capasso - Geronikaki A. - Supuran C.T.
Pharmaceuticals

Selective inhibition of helicobacter pylori carbonic anhydrases by carvacrol and thymol could impair biofilm production and the release of outer membrane vesicles

- Grande R. - Carradori S. - Puca V. - Vitale I. - Andrea Angeli - Nocentini Alessio - Bonardi A. - Gratteri P. - Lanuti P. - Bologna G. - Simeone P. - Clemente Capasso - De Luca V. - Supuran C.T.
International Journal of Molecular Sciences

Phenols from Origanum dictamnus L. and Thymus vulgaris L. and their activity against Malassezia globosa carbonic anhydrase

- Paloukopoulou C. - Govari S. - Soulioti A. - Stefanis I. - Andrea Angeli - Matheeussen A. - Clemente Capasso - Cos P. - Supuran C.T. - Karioti A.
Natural Product Research

2020

Design, synthesis, and biological evaluation of selective hCA IX inhibitors

- Carta F. - Daniela Vullo - Andrea Angeli
pH-Interfering Agents as Chemosensitizers in Cancer Therapy

Evaluation of thio-and seleno-acetamides bearing benzenesulfonamide as inhibitor of carbonic anhydrases from different pathogenic bacteria

- Andrea Angeli - Pinteala M. - Maier S.S. - Simionescu B.C. - Milaneschi A. - Abbas G. - Del Prete S. - Clemente Capasso - Capperucci A. - Tanini D. - Carta F. - Supuran C.T.
International Journal of Molecular Sciences

Crystal structure of a tetrameric type II β-carbonic anhydrase from the pathogenic bacterium burkholderia pseudomallei

- Andrea Angeli - Ferraroni M. - Pinteala M. - Maier S.S. - Simionescu B.C. - Carta F. - Del Prete S. - Clemente Capasso - Supuran C.T.
Molecules

Carbonic anhydrase inhibitors targeting metabolism and tumor microenvironment

- Andrea Angeli - Carta F. - Nocentini Alessio - Winum J.Y. - Zalubovskis R. - Akdemir A. - Onnis V. - Eldehna W.M. - Clemente Capasso - Simone G.D. - Monti S.M. - Carradori S. - Donald W.A. - Dedhar S. - Supuran C.T.
Metabolites

Benzylaminoethyureido-tailed benzenesulfonamides: Design, synthesis, kinetic and X-ray investigations on human carbonic anhydrases

- Ali M. - Murat Bozdag - Farooq U. - Andrea Angeli - Carta F. - Berto P. - Zanotti G. - Supuran C.T.
International Journal of Molecular Sciences